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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T72274 | IACS-9571 hydrochloride | ASIS-P040 hydrochloride | |
IACS-9571 (ASIS-P040) hydrochloride is a potent, selective inhibitor of TRIM24 and BRPF1, demonstrating an IC50 of 8 nM for TRIM24, and dissociation constants (Kd) of 31 nM and 14 nM for TRIM24 and BRPF1, respectively. | |||
T11597L | IACS-9571 Hydrochloride (1800477-30-8 free base) | IACS-9571 Hydrochloride,ASIS-P040 Hydrochloride | Epigenetic Reader Domain |
IACS-9571 Hydrochloride is a selective and potent inhibitor of TRIM24 and BRPF1, (IC50: 8 nM for TRIM24; Kds: 31 nM and 14 nM for TRIM24 and BRPF1). |